| Reaction Details |
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 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 3 |
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| Ligand | BDBM50647 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | uHTS absorbance assay for the identification of compounds that inhibit VHR1. |
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| IC50 | 980±n/a nM |
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| Citation |  PubChem, PC uHTS absorbance assay for the identification of compounds that inhibit VHR1. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Dual specificity protein phosphatase 3 |
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| Name: | Dual specificity protein phosphatase 3 |
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| Synonyms: | DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR |
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| Type: | Hydrolase |
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| Mol. Mass.: | 20480.58 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 185 |
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| Sequence: | MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
|
|
|
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| BDBM50647 |
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| n/a |
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| Name | BDBM50647 |
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| Synonyms: | 2,3,4,5-tetrahydroxy-6-benzo[7]annulenone | 2,3,4,5-tetrahydroxybenzo[7]annulen-6-one | 2,3,4,5-tetrahydroxybenzocyclohepten-6-one | 2,3,4,5-tetrakis(oxidanyl)benzo[7]annulen-6-one | MLS000738105 | SMR000393869 | cid_5281571 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H8O5 |
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| Mol. Mass. | 220.1782 |
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| SMILES | Oc1cc2cccc(=O)c(O)c2c(O)c1O |
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| Structure | 
|
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