Reaction Details |
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Target | Dual specificity protein phosphatase 3 |
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Ligand | BDBM51788 |
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Substrate/Competitor | n/a |
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Meas. Tech. | uHTS absorbance assay for the identification of compounds that inhibit VHR1. |
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IC50 | 2280±n/a nM |
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Citation | PubChem, PC uHTS absorbance assay for the identification of compounds that inhibit VHR1. PubChem Bioassay(2009)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Dual specificity protein phosphatase 3 |
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Name: | Dual specificity protein phosphatase 3 |
Synonyms: | DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR |
Type: | Hydrolase |
Mol. Mass.: | 20480.58 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 185 |
Sequence: | MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
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BDBM51788 |
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n/a |
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Name | BDBM51788 |
Synonyms: | 5-[(2E)-2-(8-oxidanylidenequinolin-5-ylidene)hydrazinyl]naphthalene-1-sulfonic acid | 5-[(2E)-2-(8-oxo-5-quinolinylidene)hydrazinyl]-1-naphthalenesulfonic acid | 5-[(2E)-2-(8-oxoquinolin-5-ylidene)hydrazinyl]naphthalene-1-sulfonic acid | 5-[(E)-(8-hydroxyquinolin-5-yl)diazenyl]naphthalene-1-sulfonic acid | 5-[(N'E)-N'-(8-keto-5-quinolylidene)hydrazino]naphthalene-1-sulfonic acid | MLS001197249 | SMR000555383 | cid_5876309 |
Type | Small organic molecule |
Emp. Form. | C19H13N3O4S |
Mol. Mass. | 379.389 |
SMILES | Oc1ccc(N=Nc2cccc3c(cccc23)S(O)(=O)=O)c2cccnc12 |w:6.6| |
Structure |
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