| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 55 |
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| Ligand | BDBM61011 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Image-based HTS for Selective Agonists of GPR55 |
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| EC50 | 32000±n/a nM |
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| Citation |  PubChem, PC Image-based HTS for Selective Agonists of GPR55 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G-protein coupled receptor 55 |
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| Name: | G-protein coupled receptor 55 |
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| Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36649.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1292265 |
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| Residue: | 319 |
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| Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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| BDBM61011 |
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| n/a |
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| Name | BDBM61011 |
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| Synonyms: | (3'S,4'R)-1'-(4-chlorophenyl)-2'-cyano-spiro[fluorene-9,5'-pyrazolidine]-3',4'-dicarboxylic acid dimethyl ester | (3'S,4'R)-1'-(4-chlorophenyl)-2'-cyanospiro[fluorene-9,5'-pyrazolidine]-3',4'-dicarboxylic acid dimethyl ester | MLS000549148 | SMR000113936 | cid_9499902 | dimethyl (3'S,4'R)-1'-(4-chlorophenyl)-2'-cyano-spiro[fluorene-9,5'-pyrazolidine]-3',4'-dicarboxylate | dimethyl (3'S,4'R)-1'-(4-chlorophenyl)-2'-cyanospiro[fluorene-9,5'-pyrazolidine]-3',4'-dicarboxylate | dimethyl 1-(4-chlorophenyl)-2-cyanospiro[pyrazolidine-5,9'-(9'H)-fluorene]-3,4-dicarboxylate |
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| Type | Small organic molecule |
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| Emp. Form. | C26H20ClN3O4 |
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| Mol. Mass. | 473.908 |
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| SMILES | COC(=O)[C@@H]1[C@@H](C(=O)OC)C2(N(N1C#N)c1ccc(Cl)cc1)c1ccccc1-c1ccccc21 |
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| Structure | 
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