| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 55 |
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| Ligand | BDBM61015 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Image-based HTS for Selective Agonists of GPR55 |
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| EC50 | 921.1336±n/a nM |
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| Citation |  PubChem, PC Image-based HTS for Selective Agonists of GPR55 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G-protein coupled receptor 55 |
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| Name: | G-protein coupled receptor 55 |
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| Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36649.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1292265 |
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| Residue: | 319 |
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| Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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| BDBM61015 |
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| n/a |
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| Name | BDBM61015 |
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| Synonyms: | 3-(4-fluorophenyl)-7,8-dimethoxy-5-(phenylmethyl)pyrazolo[4,3-c]quinoline | 5-benzyl-3-(4-fluorophenyl)-7,8-dimethoxy-pyrazolo[4,3-c]quinoline | 5-benzyl-3-(4-fluorophenyl)-7,8-dimethoxypyrazolo[4,3-c]quinoline | MLS000530082 | SMR000127107 | cid_2136878 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H20FN3O2 |
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| Mol. Mass. | 413.4436 |
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| SMILES | COc1cc2n(Cc3ccccc3)cc3c(nnc3c2cc1OC)-c1ccc(F)cc1 |
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| Structure | 
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