| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 55 |
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| Ligand | BDBM61021 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Image-based HTS for Selective Agonists of GPR55 |
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| EC50 | 3679.027±n/a nM |
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| Citation |  PubChem, PC Image-based HTS for Selective Agonists of GPR55 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G-protein coupled receptor 55 |
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| Name: | G-protein coupled receptor 55 |
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| Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36649.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1292265 |
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| Residue: | 319 |
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| Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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| BDBM61021 |
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| n/a |
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| Name | BDBM61021 |
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| Synonyms: | MLS000551367 | N-[2-(4-p-toluoylpiperazino)acenaphthen-1-yl]benzenesulfonamide | N-[2-[4-(4-methylbenzoyl)piperazin-1-yl]-1,2-dihydroacenaphthylen-1-yl]benzenesulfonamide | N-[2-[4-(4-methylphenyl)carbonylpiperazin-1-yl]-1,2-dihydroacenaphthylen-1-yl]benzenesulfonamide | N-[2-[4-[(4-methylphenyl)-oxomethyl]-1-piperazinyl]-1,2-dihydroacenaphthylen-1-yl]benzenesulfonamide | N-{2-[4-(4-Methyl-benzoyl)-piperazin-1-yl]-acenaphthen-1-yl}-benzenesulfonamide | SMR000145292 | cid_3540854 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H29N3O3S |
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| Mol. Mass. | 511.635 |
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| SMILES | Cc1ccc(cc1)C(=O)N1CCN(CC1)C1C(NS(=O)(=O)c2ccccc2)c2cccc3cccc1c23 |
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| Structure | 
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