Ki Summary

Reaction Details

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Target

Neuropeptide Y receptor type 2

Ligand

BDBM57782

Substrate/Competitor

n/a

Meas. Tech.

Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2.

EC50

18444±n/a nM

Citation

PubChem, PC Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Neuropeptide Y receptor type 2

Name:

Neuropeptide Y receptor type 2

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

42734.65

Organism:

Homo sapiens (Human)

Description:

NPY-Y2 NPY2R HUMAN::P49146

Residue:

381

Sequence:

MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV

BDBM57782

n/a

Name

BDBM57782

Synonyms:

4-[(3-allyl-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)methyl]-2-ethoxy-3-nitrophenyl acetate | MLS000663880 | SMR000292408 | [2-ethoxy-3-nitro-4-[(Z)-(4-oxidanylidene-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]phenyl] ethanoate | [2-ethoxy-3-nitro-4-[(Z)-(4-oxo-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]phenyl] acetate | acetic acid [2-ethoxy-3-nitro-4-[(Z)-(4-oxo-3-prop-2-enyl-2-sulfanylidene-5-thiazolidinylidene)methyl]phenyl] ester | acetic acid [4-[(Z)-(3-allyl-4-keto-2-thioxo-thiazolidin-5-ylidene)methyl]-2-ethoxy-3-nitro-phenyl] ester | cid_2191297

Type

Small organic molecule

Emp. Form.

C17H16N2O6S2

Mol. Mass.

408.449

SMILES

CCOc1c(OC(C)=O)ccc(\C=C2/SC(=S)N(CC=C)C2=O)c1[N+]([O-])=O

Structure