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TargetNeuropeptide Y receptor type 2
LigandBDBM58193
Substrate/Competitorn/a
Meas. Tech.Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2.
EC50 8237±n/a nM
Citation PubChem, PC Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Neuropeptide Y receptor type 2
Name:Neuropeptide Y receptor type 2
Synonyms:NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:Enzyme Catalytic Domain
Mol. Mass.:42734.65
Organism:Homo sapiens (Human)
Description:NPY-Y2 NPY2R HUMAN::P49146
Residue:381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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  Blast E-value cutoff:
BDBM58193
n/a
NameBDBM58193
Synonyms:1-(3,4-dichlorophenyl)-3-[2-[2,6-dinitro-4-(trifluoromethyl)anilino]ethyl]thiourea | 1-(3,4-dichlorophenyl)-3-[2-[[2,6-dinitro-4-(trifluoromethyl)phenyl]amino]ethyl]thiourea | MLS000833819 | N-(3,4-dichlorophenyl)-N'-{2-[2,6-dinitro-4-(trifluoromethyl)anilino]ethyl}thiourea | SMR000457540 | cid_2803877
TypeSmall organic molecule
Emp. Form.C16H12Cl2F3N5O4S
Mol. Mass.498.264
SMILES[O-][N+](=O)c1cc(cc(c1NCCNC(=S)Nc1ccc(Cl)c(Cl)c1)[N+]([O-])=O)C(F)(F)F
Structure
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