Reaction Details |
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Target | Regulator of G-protein signaling 4 |
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Ligand | BDBM47734 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds |
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EC50 | 6607±n/a nM |
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Citation | PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds PubChem Bioassay(2010)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Regulator of G-protein signaling 4 |
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Name: | Regulator of G-protein signaling 4 |
Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
Type: | Enzyme |
Mol. Mass.: | 23263.51 |
Organism: | Homo sapiens (Human) |
Description: | P49798 |
Residue: | 205 |
Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM47734 |
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n/a |
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Name | BDBM47734 |
Synonyms: | MLS000553854 | N-[(4-methylphenyl)-(5-nitro-8-oxidanyl-quinolin-7-yl)methyl]propanamide | N-[(8-Hydroxy-5-nitro-quinolin-7-yl)-p-tolyl-methyl]-propionamide | N-[(8-hydroxy-5-nitro-7-quinolinyl)-(4-methylphenyl)methyl]propanamide | N-[(8-hydroxy-5-nitro-7-quinolyl)-(p-tolyl)methyl]propionamide | N-[(8-hydroxy-5-nitroquinolin-7-yl)-(4-methylphenyl)methyl]propanamide | SMR000172089 | cid_2922056 |
Type | Small organic molecule |
Emp. Form. | C20H19N3O4 |
Mol. Mass. | 365.3826 |
SMILES | CCC(=O)NC(c1ccc(C)cc1)c1cc([N+]([O-])=O)c2cccnc2c1O |
Structure |
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