| Reaction Details |
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 | Report a problem with these data |
| Target | Regulator of G-protein signaling 4 |
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| Ligand | BDBM47798 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds |
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| EC50 | 30000±n/a nM |
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| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Regulator of G-protein signaling 4 |
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| Name: | Regulator of G-protein signaling 4 |
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| Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 23263.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49798 |
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| Residue: | 205 |
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| Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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| BDBM47798 |
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| n/a |
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| Name | BDBM47798 |
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| Synonyms: | 4-chloranyl-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl-N-methyl-1,3,5-triazin-2-amine | 4-chloro-6-(4,6-dimethylpyrimidin-2-yl)sulfanyl-N-methyl-1,3,5-triazin-2-amine | 4-chloro-6-[(4,6-dimethyl-2-pyrimidinyl)thio]-N-methyl-1,3,5-triazin-2-amine | MLS000707335 | SMR000288800 | [4-chloro-6-[(4,6-dimethylpyrimidin-2-yl)thio]-s-triazin-2-yl]-methyl-amine | cid_1087037 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H11ClN6S |
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| Mol. Mass. | 282.753 |
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| SMILES | CNc1nc(Cl)nc(Sc2nc(C)cc(C)n2)n1 |
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| Structure | 
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