| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM54798 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | HTS Image-Based Screen for Antagonists of the DOR Receptor |
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| IC50 | 23446±n/a nM |
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| Citation |  PubChem, PC HTS Image-Based Screen for Antagonists of the DOR Receptor PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40382.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. |
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| Residue: | 372 |
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| Sequence: | MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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|
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| BDBM54798 |
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| n/a |
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| Name | BDBM54798 |
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| Synonyms: | (5Z)-2-azanylidene-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-(1,3-thiazol-2-yl)-1,3-thiazolidin-4-one | (5Z)-2-imino-5-[(2-methyl-1H-indol-3-yl)methylene]-3-thiazol-2-yl-thiazolidin-4-one | (5Z)-2-imino-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-(1,3-thiazol-2-yl)-1,3-thiazolidin-4-one | (5Z)-2-imino-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-(2-thiazolyl)-4-thiazolidinone | MLS000519510 | SMR000129929 | cid_5291664 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H12N4OS2 |
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| Mol. Mass. | 340.423 |
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| SMILES | Cc1[nH]c2ccccc2c1\C=C1/SC(=N)N(C1=O)c1nccs1 |
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| Structure | 
|
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