| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM54799 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | HTS Image-Based Screen for Antagonists of the DOR Receptor |
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| IC50 | 10658±n/a nM |
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| Citation |  PubChem, PC HTS Image-Based Screen for Antagonists of the DOR Receptor PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40382.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. |
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| Residue: | 372 |
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| Sequence: | MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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|
|
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| BDBM54799 |
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| n/a |
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| Name | BDBM54799 |
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| Synonyms: | 2-(2,3,4,5,6-pentafluorophenyl)-1-benzopyran-4-one | 2-(2,3,4,5,6-pentafluorophenyl)chromen-4-one | 2-(2,3,4,5,6-pentafluorophenyl)chromone | 2-[2,3,4,5,6-pentakis(fluoranyl)phenyl]chromen-4-one | MLS000568955 | SMR000149965 | cid_2055076 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H5F5O2 |
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| Mol. Mass. | 312.191 |
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| SMILES | Fc1c(F)c(F)c(c(F)c1F)-c1cc(=O)c2ccccc2o1 |
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| Structure | 
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