Ki Summary

Reaction Details

Report a problem with these data

Target

Trans-activator protein BZLF1

Ligand

BDBM62492

Substrate/Competitor

n/a

Meas. Tech.

Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA

IC50

111248±n/a nM

Citation

PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Trans-activator protein BZLF1

Name:

Trans-activator protein BZLF1

Synonyms:

BZLF1 | BZLF1_EBVB9 | PPP5C protein

Type:

Enzyme Catalytic Domain

Mol. Mass.:

26856.37

Organism:

Human herpesvirus 4

Description:

gi_82503229

Residue:

245

Sequence:

MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQ
LTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNS
TVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRY
KNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHE
DLLNF

BDBM62492

n/a

Name

BDBM62492

Synonyms:

2-[(5Z)-2,4-bis(oxidanylidene)-5-[(2,4,6-trimethoxyphenyl)methylidene]-1,3-thiazolidin-3-yl]-N-(2-fluorophenyl)ethanamide | 2-[(5Z)-2,4-diketo-5-(2,4,6-trimethoxybenzylidene)thiazolidin-3-yl]-N-(2-fluorophenyl)acetamide | 2-[(5Z)-2,4-dioxo-5-[(2,4,6-trimethoxyphenyl)methylidene]-1,3-thiazolidin-3-yl]-N-(2-fluorophenyl)acetamide | 2-[(5Z)-2,4-dioxo-5-[(2,4,6-trimethoxyphenyl)methylidene]-3-thiazolidinyl]-N-(2-fluorophenyl)acetamide | 2-[2,4-dioxo-5-(2,4,6-trimethoxybenzylidene)-1,3-thiazolidin-3-yl]-N-(2-fluorophenyl)acetamide | MLS001180205 | SMR000477449 | cid_1231499

Type

Small organic molecule

Emp. Form.

C21H19FN2O6S

Mol. Mass.

446.449

SMILES

COc1cc(OC)c(\C=C2/SC(=O)N(CC(=O)Nc3ccccc3F)C2=O)c(OC)c1

Structure