| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Heat shock factor protein 1 |
|---|
| Ligand | BDBM3789 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Luminescence Cell-Based Dose Confimation HTS to Identify Inhibitors of Heat Shock Factor 1 (HSF1) |
|---|
| EC50 | >195000±0 nM |
|---|
| Citation |  PubChem, PC Luminescence Cell-Based Dose Confimation HTS to Identify Inhibitors of Heat Shock Factor 1 (HSF1) PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Heat shock factor protein 1 |
|---|
| Name: | Heat shock factor protein 1 |
|---|
| Synonyms: | HSF1_MOUSE | Hsf1 | Hsf1 protein |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 57208.68 |
|---|
| Organism: | Mus musculus |
|---|
| Description: | P38532 |
|---|
| Residue: | 525 |
|---|
| Sequence: | MDLAVGPGAAGPSNVPAFLTKLWTLVSDPDTDALICWSPSGNSFHVFDQGQFAKEVLPKY
FKHNNMASFVRQLNMYGFRKVVHIEQGGLVKPERDDTEFQHPCFLRGQEQLLENIKRKVT
SVSTLKSEDIKIRQDSVTRLLTDVQLMKGKQECMDSKLLAMKHENEALWREVASLRQKHA
QQQKVVNKLIQFLISLVQSNRILGVKRKIPLMLSDSNSAHSVPKYGRQYSLEHVHGPGPY
SAPSPAYSSSSLYSSDAVTSSGPIISDITELAPTSPLASPGRSIDERPLSSSTLVRVKQE
PPSPPHSPRVLEASPGRPSSMDTPLSPTAFIDSILRESEPTPAASNTAPMDTTGAQAPAL
PTPSTPEKCLSVACLDKNELSDHLDAMDSNLDNLQTMLTSHGFSVDTSALLDLFSPSVTM
PDMSLPDLDSSLASIQELLSPQEPPRPIEAENSNPDSGKQLVHYTAQPLFLLDPDAVDTG
SSELPVLFELGESSYFSEGDDYTDDPTISLLTGTEPHKAKDPTVS
|
|
|
|---|
| BDBM3789 |
|---|
| n/a |
|---|
| Name | BDBM3789 |
|---|
| Synonyms: | 1-Phenylbenzimidazole Analog 6 | 2-phenyl-1H-1,3-benzodiazole | US9138393, 2-Phenyl benzimidazole | US9144538, 2-Phenyl benzimidazole | cid_12855 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C13H10N2 |
|---|
| Mol. Mass. | 194.2319 |
|---|
| SMILES | c1ccc(cc1)-c1nc2ccccc2[nH]1 |
|---|
| Structure | 
|
|---|
Search and Browse
