| Reaction Details |
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 | Report a problem with these data |
| Target | Photoreceptor-specific nuclear receptor |
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| Ligand | BDBM66212 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3) |
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| IC50 | >39841±n/a nM |
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| Citation |  PubChem, PC TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3) PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Photoreceptor-specific nuclear receptor |
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| Name: | Photoreceptor-specific nuclear receptor |
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| Synonyms: | NR2E3 | NR2E3_HUMAN | PNR | RNR | photoreceptor-specific nuclear receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 44699.83 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_401901 |
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| Residue: | 410 |
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| Sequence: | METRPTALMSSTVAAAAPAAGAASRKESPGRWGLGEDPTGVSPSLQCRVCGDSSSGKHYG
IYACNGCSGFFKRSVRRRLIYRCQVGAGMCPVDKAHRNQCQACRLKKCLQAGMNQDAVQN
ERQPRSTAQVHLDSMESNTESRPESLVAPPAPAGRSPRGPTPMSAARALGHHFMASLITA
ETCAKLEPEDADENIDVTSNDPEFPSSPYSSSSPCGLDSIHETSARLLFMAVKWAKNLPV
FSSLPFRDQVILLEEAWSELFLLGAIQWSLPLDSCPLLAPPEASAAGGAQGRLTLASMET
RVLQETISRFRALAVDPTEFACMKALVLFKPETRGLKDPEHVEALQDQSQVMLSQHSKAH
HPSQPVRFGKLLLLLPSLRFITAERIELLFFRKTIGNTPMEKLLCDMFKN
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| BDBM66212 |
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| n/a |
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| Name | BDBM66212 |
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| Synonyms: | 3-[(7-methoxy-1-benzofuran-2-yl)carbonyl]-1-(5-methyl-1,2-oxazol-3-yl)-4-oxidanyl-2-thiophen-2-yl-2H-pyrrol-5-one | 3-hydroxy-4-(7-methoxybenzofuran-2-carbonyl)-1-(5-methylisoxazol-3-yl)-5-(2-thienyl)-3-pyrrolin-2-one | 4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-1-(5-methyl-1,2-oxazol-3-yl)-2-thiophen-2-yl-2H-pyrrol-5-one | 4-hydroxy-3-[(7-methoxy-2-benzofuranyl)-oxomethyl]-1-(5-methyl-3-isoxazolyl)-2-thiophen-2-yl-2H-pyrrol-5-one | MLS001125423 | SMR000668743 | cid_2964736 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H16N2O6S |
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| Mol. Mass. | 436.437 |
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| SMILES | COc1cccc2cc(oc12)C(=O)C1C(N(C(=O)C1=O)c1cc(C)on1)c1cccs1 |
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| Structure | 
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