| Reaction Details |
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 | Report a problem with these data |
| Target | DNA damage-inducible transcript 3 protein |
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| Ligand | BDBM68017 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose-response primary assay and counterscreen assay for HTS small molecule inhibitors of CHOP to regulate the unfolded protein response to ER stress |
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| IC50 | 360±n/a nM |
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| Citation |  PubChem, PC Dose-response primary assay and counterscreen assay for HTS small molecule inhibitors of CHOP to regulate the unfolded protein response to ER stress PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| DNA damage-inducible transcript 3 protein |
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| Name: | DNA damage-inducible transcript 3 protein |
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| Synonyms: | Chop | Chop10 | DDIT3_MOUSE | Ddit3 | Gadd153 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 19175.17 |
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| Organism: | Mus musculus |
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| Description: | gi_160707929 |
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| Residue: | 168 |
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| Sequence: | MAAESLPFTLETVSSWELEAWYEDLQEVLSSDEIGGTYISSPGNEEEESKTFTTLDPASL
AWLTEEPGPTEVTRTSQSPRSPDSSQSSMAQEEEEEEQGRTRKRKQSGQCPARPGKQRMK
EKEQENERKVAQLAEENERLKQEIERLTREVETTRRALIDRMVSLHQA
|
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| BDBM68017 |
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| n/a |
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| Name | BDBM68017 |
|---|
| Synonyms: | 2-(4-methylanilino)-N-[(3-phenoxyphenyl)methylideneamino]acetamide | 2-[(4-methylphenyl)amino]-N'-[(1E)-(3-phenoxyphenyl)methylene]acetohydrazide | 2-[(4-methylphenyl)amino]-N-[(3-phenoxyphenyl)methylideneamino]ethanamide | MLS000586151 | N-[(3-phenoxybenzylidene)amino]-2-(p-toluidino)acetamide | SMR000204514 | cid_1520328 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H21N3O2 |
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| Mol. Mass. | 359.421 |
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| SMILES | Cc1ccc(NCC(=O)NN=Cc2cccc(Oc3ccccc3)c2)cc1 |
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| Structure | 
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