Ki Summary

Reaction Details

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Target

Cannabinoid receptor 2

Ligand

BDBM68309

Substrate/Competitor

n/a

Meas. Tech.

SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2

IC50

>32000±n/a nM

Citation

PubChem, PC SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Cannabinoid receptor 2

Name:

Cannabinoid receptor 2

Synonyms:

CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2

Type:

G Protein-Coupled Receptor (GPCR)

Mol. Mass.:

39690.94

Organism:

Homo sapiens (Human)

Description:

P34972

Residue:

360

Sequence:

MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC

BDBM68309

n/a

Name

BDBM68309

Synonyms:

MLS-0435535.0001 | N-(2-methoxy-5-morpholin-4-ylsulfonyl-phenyl)-5-methyl-4-propyl-thiophene-2-carboxamide | N-(2-methoxy-5-morpholin-4-ylsulfonylphenyl)-5-methyl-4-propylthiophene-2-carboxamide | N-(2-methoxy-5-morpholinosulfonyl-phenyl)-5-methyl-4-propyl-thiophene-2-carboxamide | N-[2-methoxy-5-(4-morpholinylsulfonyl)phenyl]-5-methyl-4-propyl-2-thiophenecarboxamide | cid_16279444

Type

Small organic molecule

Emp. Form.

C20H26N2O5S2

Mol. Mass.

438.561

SMILES

CCCc1cc(sc1C)C(=O)Nc1cc(ccc1OC)S(=O)(=O)N1CCOCC1

Structure