| Reaction Details |
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 | Report a problem with these data |
| Target | Protein Rev |
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| Ligand | BDBM32120 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction |
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| IC50 | 19371±n/a nM |
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| Citation |  PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Protein Rev |
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| Name: | Protein Rev |
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| Synonyms: | Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev |
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| Type: | PROTEIN |
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| Mol. Mass.: | 13078.11 |
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| Organism: | Human immunodeficiency virus 1 |
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| Description: | ChEMBL_79479 |
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| Residue: | 116 |
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| Sequence: | MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERIL
GTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
|
|
|
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| BDBM32120 |
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| n/a |
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| Name | BDBM32120 |
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| Synonyms: | 2-[[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfinyl]-N-(pyridin-2-ylmethyl)acetamide | 2-[[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfinyl]-N-(pyridin-2-ylmethyl)ethanamide | 2-[[2-(4-methoxyphenyl)-5-methyl-4-oxazolyl]methylsulfinyl]-N-(2-pyridinylmethyl)acetamide | 2-[[2-(4-methoxyphenyl)-5-methyl-oxazol-4-yl]methylsulfinyl]-N-(2-pyridylmethyl)acetamide | MLS000117623 | SMR000094571 | cid_5308158 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H21N3O4S |
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| Mol. Mass. | 399.463 |
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| SMILES | COc1ccc(cc1)-c1nc(CS(=O)CC(=O)NCc2ccccn2)c(C)o1 |
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| Structure | 
|
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