| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Heat shock factor protein 1 |
|---|
| Ligand | BDBM37386 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Luminescence Cell-Based Dose Retest to Identify Potentiators of Heat Shock Factor 1 (HSF1) |
|---|
| EC50 | >260000±n/a nM |
|---|
| Citation |  PubChem, PC Luminescence Cell-Based Dose Retest to Identify Potentiators of Heat Shock Factor 1 (HSF1) PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Heat shock factor protein 1 |
|---|
| Name: | Heat shock factor protein 1 |
|---|
| Synonyms: | HSF1_MOUSE | Hsf1 | Hsf1 protein |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 57208.68 |
|---|
| Organism: | Mus musculus |
|---|
| Description: | P38532 |
|---|
| Residue: | 525 |
|---|
| Sequence: | MDLAVGPGAAGPSNVPAFLTKLWTLVSDPDTDALICWSPSGNSFHVFDQGQFAKEVLPKY
FKHNNMASFVRQLNMYGFRKVVHIEQGGLVKPERDDTEFQHPCFLRGQEQLLENIKRKVT
SVSTLKSEDIKIRQDSVTRLLTDVQLMKGKQECMDSKLLAMKHENEALWREVASLRQKHA
QQQKVVNKLIQFLISLVQSNRILGVKRKIPLMLSDSNSAHSVPKYGRQYSLEHVHGPGPY
SAPSPAYSSSSLYSSDAVTSSGPIISDITELAPTSPLASPGRSIDERPLSSSTLVRVKQE
PPSPPHSPRVLEASPGRPSSMDTPLSPTAFIDSILRESEPTPAASNTAPMDTTGAQAPAL
PTPSTPEKCLSVACLDKNELSDHLDAMDSNLDNLQTMLTSHGFSVDTSALLDLFSPSVTM
PDMSLPDLDSSLASIQELLSPQEPPRPIEAENSNPDSGKQLVHYTAQPLFLLDPDAVDTG
SSELPVLFELGESSYFSEGDDYTDDPTISLLTGTEPHKAKDPTVS
|
|
|
|---|
| BDBM37386 |
|---|
| n/a |
|---|
| Name | BDBM37386 |
|---|
| Synonyms: | 2-keto-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazol[4,3-a]azepin-3-yl)phenyl]-3H-1,3-benzoxazole-6-sulfonamide | 2-oxidanylidene-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-3H-1,3-benzoxazole-6-sulfonamide | 2-oxo-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-3H-1,3-benzoxazole-6-sulfonamide | MLS000053769 | SMR000068222 | cid_2997804 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H19N5O4S |
|---|
| Mol. Mass. | 425.461 |
|---|
| SMILES | O=c1[nH]c2ccc(cc2o1)S(=O)(=O)Nc1ccc(cc1)-c1nnc2CCCCCn12 |
|---|
| Structure | 
|
|---|
Search and Browse
