| Reaction Details |
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 | Report a problem with these data |
| Target | G protein-activated inward rectifier potassium channel 1 |
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| Ligand | BDBM10759 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Measurement of GPCR-mediated thallium flux through GIRK channels: Dose-Response Testing |
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| EC50 | 0.06142±n/a nM |
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| Citation |  PubChem, PC Measurement of GPCR-mediated thallium flux through GIRK channels: Dose-Response Testing PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G protein-activated inward rectifier potassium channel 1 |
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| Name: | G protein-activated inward rectifier potassium channel 1 |
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| Synonyms: | Girk1 | KCNJ3_RAT | Kcnj3 | Kga |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 56581.73 |
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| Organism: | Rattus norvegicus |
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| Description: | gi_13928834 |
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| Residue: | 501 |
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| Sequence: | MSALRRKFGDDYQVVTTSSSGSGLQPQGPGQGPQQQLVPKKKRQRFVDKNGRCNVQHGNL
GSETSRYLSDLFTTLVDLKWRWNLFIFILTYTVAWLFMASMWWVIAYTRGDLNKAHVGNY
TPCVANVYNFPSAFLFFIETEATIGYGYRYITDKCPEGIILFLFQSILGSIVDAFLIGCM
FIKMSQPKKRAETLMFSEHAVISMRDGKLTLMFRVGNLRNSHMVSAQIRCKLLKSRQTPE
GEFLPLDQLELDVGFSTGADQLFLVSPLTICHVIDAKSPFYDLSQRSMQTEQFEVVVILE
GIVETTGMTCQARTSYTEDEVLWGHRFFPVISLEEGFFKVDYSQFHATFEVPTPPYSVKE
QEEMLLMSSPLIAPAITNSKERHNSVECLDGLDDISTKLPSKLQKITGREDFPKKLLRMS
STTSEKAYSLGDLPMKLQRISSVPGNSEEKLVSKTTKMLSDPMSQSVADLPPKLQKMAGG
PTRMEGNLPAKLRKMNSDRFT
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| BDBM10759 |
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| n/a |
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| Name | BDBM10759 |
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| Synonyms: | 2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acetoxyethyl(trimethyl)ammonium;perchlorate | CHEMBL667 | US10667515, Compound ACh | [2-(acetyloxy)ethyl]trimethylazanium | acetylcholine | acetylcholine chloride | cid_6060 |
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| Type | Small Organic Molecule |
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| Emp. Form. | C7H16NO2 |
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| Mol. Mass. | 146.2069 |
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| SMILES | CC(=O)OCC[N+](C)(C)C |
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| Structure | 
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