Reaction Details | |||
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Target | Protein LANA1 | ||
Ligand | BDBM74308 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | Fluorescence Polarization Cell-Free Homogeneous Dose Retest to Confirm Inhibitors of the LANA Histone H2A/H2B Interaction | ||
EC50 | >75000±n/a nM | ||
Citation | PubChem, PC Fluorescence Polarization Cell-Free Homogeneous Dose Retest to Confirm Inhibitors of the LANA Histone H2A/H2B Interaction PubChem Bioassay(2010)[AID] | ||
More Info.: | Get all data from this article, Solution Info, Assay Method | ||
Protein LANA1 | |||
Name: | Protein LANA1 | ||
Synonyms: | LANA | LANA1 | LANA1_HHV8P | ||
Type: | Enzyme Catalytic Domain | ||
Mol. Mass.: | 131093.36 | ||
Organism: | Human herpesvirus 8 | ||
Description: | Q9QR71 | ||
Residue: | 1129 | ||
Sequence: |
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BDBM74308 | |||
n/a | |||
Name | BDBM74308 | ||
Synonyms: | 4-[(3-nitrophenyl)sulfonylamino]-N-(4-oxidanylcyclohexyl)benzamide | MLS002180713 | N-(4-hydroxycyclohexyl)-4-[(3-nitrophenyl)sulfonylamino]benzamide | SMR001269743 | cid_25162777 | ||
Type | Small organic molecule | ||
Emp. Form. | C19H21N3O6S | ||
Mol. Mass. | 419.452 | ||
SMILES | OC1CCC(CC1)NC(=O)c1ccc(NS(=O)(=O)c2cccc(c2)[N+]([O-])=O)cc1 |(4.41,-8.23,;4.41,-6.69,;5.75,-5.92,;5.75,-4.38,;4.41,-3.61,;3.08,-4.38,;3.08,-5.92,;4.41,-2.07,;5.75,-1.3,;7.08,-2.07,;5.75,.24,;4.41,1.01,;4.41,2.55,;5.75,3.32,;5.75,4.86,;7.08,5.63,;6.31,6.96,;7.85,4.3,;8.41,6.4,;8.41,7.94,;9.75,8.71,;11.08,7.94,;11.08,6.4,;9.75,5.63,;12.42,5.63,;13.75,6.4,;12.42,4.09,;7.08,2.55,;7.08,1.01,)| | ||
Structure |