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TargetTyrosine-protein phosphatase non-receptor type 7
LigandBDBM74519
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2
IC50>79400±0 nM
Citation PubChem, PC Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2 PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Tyrosine-protein phosphatase non-receptor type 7
Name:Tyrosine-protein phosphatase non-receptor type 7
Synonyms:He-PTP | Hematopoietic protein-tyrosine phosphatase | Hematopoietic protein-tyrosine phosphatase (HEPTP) | PTN7_HUMAN | PTPN7 | Protein-tyrosine phosphatase LC-PTP | Tyrosine-protein phosphatase non-receptor type 7 | Tyrosine-protein phosphatase non-receptor type 7 (HEPTP)
Type:Protein
Mol. Mass.:40530.79
Organism:Homo sapiens (Human)
Description:P35236
Residue:360
Sequence:
MVQAHGGRSRAQPLTLSLGAAMTQPPPEKTPAKKHVRLQERRGSNVALMLDVRSLGAVEP
ICSVNTPREVTLHFLRTAGHPLTRWALQRQPPSPKQLEEEFLKIPSNFVSPEDLDIPGHA
SKDRYKTILPNPQSRVCLGRAQSQEDGDYINANYIRGYDGKEKVYIATQGPMPNTVSDFW
EMVWQEEVSLIVMLTQLREGKEKCVHYWPTEEETYGPFQIRIQDMKECPEYTVRQLTIQY
QEERRSVKHILFSAWPDHQTPESAGPLLRLVAEVEESPETAAHPGPIVVHCSAGIGRTGC
FIATRIGCQQLKARGEVDILGIVCQLRLDRGGMIQTAEQYQFLHHTLALYAGQLPEEPSP
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  Blast E-value cutoff:
BDBM74519
n/a
NameBDBM74519
Synonyms:1-(4-nitrophenyl)-4-(2-thienylacetyl)piperazine | 1-[4-(4-nitrophenyl)-1-piperazinyl]-2-thiophen-2-ylethanone | 1-[4-(4-nitrophenyl)piperazin-1-yl]-2-thiophen-2-yl-ethanone | 1-[4-(4-nitrophenyl)piperazin-1-yl]-2-thiophen-2-ylethanone | 1-[4-(4-nitrophenyl)piperazino]-2-(2-thienyl)ethanone | MLS000684504 | SMR000269682 | cid_2904576
TypeSmall organic molecule
Emp. Form.C16H17N3O3S
Mol. Mass.331.389
SMILES[O-][N+](=O)c1ccc(cc1)N1CCN(CC1)C(=O)Cc1cccs1
Structure
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