| Reaction Details |
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 | Report a problem with these data |
| Target | Tyrosine-protein phosphatase non-receptor type 7 |
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| Ligand | BDBM74536 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2 |
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| IC50 | >79400±0 nM |
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| Citation |  PubChem, PC Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Tyrosine-protein phosphatase non-receptor type 7 |
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| Name: | Tyrosine-protein phosphatase non-receptor type 7 |
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| Synonyms: | He-PTP | Hematopoietic protein-tyrosine phosphatase | Hematopoietic protein-tyrosine phosphatase (HEPTP) | PTN7_HUMAN | PTPN7 | Protein-tyrosine phosphatase LC-PTP | Tyrosine-protein phosphatase non-receptor type 7 | Tyrosine-protein phosphatase non-receptor type 7 (HEPTP) |
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| Type: | Protein |
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| Mol. Mass.: | 40530.79 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35236 |
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| Residue: | 360 |
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| Sequence: | MVQAHGGRSRAQPLTLSLGAAMTQPPPEKTPAKKHVRLQERRGSNVALMLDVRSLGAVEP
ICSVNTPREVTLHFLRTAGHPLTRWALQRQPPSPKQLEEEFLKIPSNFVSPEDLDIPGHA
SKDRYKTILPNPQSRVCLGRAQSQEDGDYINANYIRGYDGKEKVYIATQGPMPNTVSDFW
EMVWQEEVSLIVMLTQLREGKEKCVHYWPTEEETYGPFQIRIQDMKECPEYTVRQLTIQY
QEERRSVKHILFSAWPDHQTPESAGPLLRLVAEVEESPETAAHPGPIVVHCSAGIGRTGC
FIATRIGCQQLKARGEVDILGIVCQLRLDRGGMIQTAEQYQFLHHTLALYAGQLPEEPSP
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| BDBM74536 |
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| n/a |
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| Name | BDBM74536 |
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| Synonyms: | 2-[3-(3-fluoranyl-4-methyl-phenyl)-2,4-bis(oxidanylidene)thieno[3,2-d]pyrimidin-1-yl]-N-(oxolan-2-ylmethyl)ethanamide | 2-[3-(3-fluoro-4-methyl-phenyl)-2,4-diketo-thieno[3,2-d]pyrimidin-1-yl]-N-(tetrahydrofurfuryl)acetamide | 2-[3-(3-fluoro-4-methylphenyl)-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]-N-(2-oxolanylmethyl)acetamide | 2-[3-(3-fluoro-4-methylphenyl)-2,4-dioxothieno[3,2-d]pyrimidin-1-yl]-N-(oxolan-2-ylmethyl)acetamide | MLS000950328 | SMR000621722 | cid_6621355 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H20FN3O4S |
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| Mol. Mass. | 417.454 |
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| SMILES | Cc1ccc(cc1F)-n1c(=O)n(CC(=O)NCC2CCCO2)c2ccsc2c1=O |
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| Structure | 
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