| Reaction Details |
|---|
 | Report a problem with these data |
| Target | G-protein coupled receptor 35 |
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| Ligand | BDBM76072 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 6 |
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| IC50 | >32000±n/a nM |
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| Citation |  PubChem, PC SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 6 PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| G-protein coupled receptor 35 |
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| Name: | G-protein coupled receptor 35 |
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| Synonyms: | G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 34085.57 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_33695097 |
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| Residue: | 309 |
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| Sequence: | MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
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|
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| BDBM76072 |
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| n/a |
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| Name | BDBM76072 |
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| Synonyms: | 4-(4-methoxyphenyl)-7-methyl-2-(4-methylphenyl)pyrazolo[3,4-d]pyridazine | 4-(4-methoxyphenyl)-7-methyl-2-(p-tolyl)pyrazolo[3,4-d]pyridazine | MLS-0437176.0001 | cid_42600928 |
|---|
| Type | Small organic molecule |
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| Emp. Form. | C20H18N4O |
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| Mol. Mass. | 330.3831 |
|---|
| SMILES | COc1ccc(cc1)-c1nnc(C)c2nn(cc12)-c1ccc(C)cc1 |
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| Structure | 
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