Reaction Details |
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Target | Mu-type opioid receptor |
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Ligand | BDBM75392 |
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Substrate/Competitor | n/a |
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Meas. Tech. | SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay - Set 3 |
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EC50 | >32000±n/a nM |
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Citation | PubChem, PC SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay - Set 3 PubChem Bioassay(2010)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Mu-type opioid receptor |
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Name: | Mu-type opioid receptor |
Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 44789.51 |
Organism: | Homo sapiens (Human) |
Description: | P35372 |
Residue: | 400 |
Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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BDBM75392 |
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n/a |
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Name | BDBM75392 |
Synonyms: | KSC-5-289E5 | KUC104196N | [4-[[5-pyridin-2-yl-4-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]phenyl] acetate | [4-[[5-pyridin-2-yl-4-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]phenyl] ethanoate | acetic acid [4-[[[5-(2-pyridinyl)-4-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]thio]methyl]phenyl] ester | acetic acid [4-[[[5-(2-pyridyl)-4-(2-thenyl)-1,2,4-triazol-3-yl]thio]methyl]phenyl] ester | cid_44620931 |
Type | Small organic molecule |
Emp. Form. | C21H18N4O2S2 |
Mol. Mass. | 422.523 |
SMILES | CC(=O)Oc1ccc(CSc2nnc(-c3ccccn3)n2Cc2cccs2)cc1 |
Structure |
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