| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Mu-type opioid receptor |
|---|
| Ligand | BDBM75393 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay - Set 3 |
|---|
| EC50 | >32000±n/a nM |
|---|
| Citation |  PubChem, PC SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay - Set 3 PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Mu-type opioid receptor |
|---|
| Name: | Mu-type opioid receptor |
|---|
| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 44789.51 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P35372 |
|---|
| Residue: | 400 |
|---|
| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
|
|
|
|---|
| BDBM75393 |
|---|
| n/a |
|---|
| Name | BDBM75393 |
|---|
| Synonyms: | 2-[5-[(4-isopropylbenzyl)thio]-4-(2-thenyl)-1,2,4-triazol-3-yl]pyridine | 2-[5-[(4-propan-2-ylphenyl)methylsulfanyl]-4-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]pyridine | 2-[5-[(4-propan-2-ylphenyl)methylthio]-4-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]pyridine | KSC-5-289F6 | KUC104197N | cid_44620929 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C22H22N4S2 |
|---|
| Mol. Mass. | 406.567 |
|---|
| SMILES | CC(C)c1ccc(CSc2nnc(-c3ccccn3)n2Cc2cccs2)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
