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TargetSentrin-specific protease 8
LigandBDBM76463
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay
IC50 7470±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sentrin-specific protease 8
Name:Sentrin-specific protease 8
Synonyms:DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8
Type:Enzyme Catalytic Domain
Mol. Mass.:24104.52
Organism:Homo sapiens (Human)
Description:gi_262118306
Residue:212
Sequence:
MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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  Blast E-value cutoff:
BDBM76463
n/a
NameBDBM76463
Synonyms:4-Methyl-5-phenyl-thiophene-3-carboxylic acid phenylamide | 4-methyl-N,5-diphenyl-3-thiophenecarboxamide | 4-methyl-N,5-diphenyl-thiophene-3-carboxamide | 4-methyl-N,5-diphenylthiophene-3-carboxamide | MLS000564604 | SMR000177122 | cid_829294
TypeSmall organic molecule
Emp. Form.C18H15NOS
Mol. Mass.293.383
SMILESCc1c(csc1-c1ccccc1)C(=O)Nc1ccccc1
Structure
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