Reaction Details |
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Target | Sentrin-specific protease 8 |
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Ligand | BDBM76564 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay |
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IC50 | 11600±n/a nM |
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Citation | PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Sentrin-specific protease 8 |
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Name: | Sentrin-specific protease 8 |
Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 24104.52 |
Organism: | Homo sapiens (Human) |
Description: | gi_262118306 |
Residue: | 212 |
Sequence: | MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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BDBM76564 |
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n/a |
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Name | BDBM76564 |
Synonyms: | (4E)-4-(ethoxymethylene)-2-(4-methoxyphenyl)isoquinoline-1,3-quinone | (4E)-4-(ethoxymethylidene)-2-(4-methoxyphenyl)isoquinoline-1,3-dione | MLS001007186 | SMR000048645 | cid_1970378 |
Type | Small organic molecule |
Emp. Form. | C19H17NO4 |
Mol. Mass. | 323.3426 |
SMILES | CCO\C=C1\C(=O)N(C(=O)c2ccccc12)c1ccc(OC)cc1 |
Structure |
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