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TargetSentrin-specific protease 8
LigandBDBM76702
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay
IC50 2410±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sentrin-specific protease 8
Name:Sentrin-specific protease 8
Synonyms:DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8
Type:Enzyme Catalytic Domain
Mol. Mass.:24104.52
Organism:Homo sapiens (Human)
Description:gi_262118306
Residue:212
Sequence:
MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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  Blast E-value cutoff:
BDBM76702
n/a
NameBDBM76702
Synonyms:MLS001193335 | N,3-diphenyl-1,2,4-thiadiazol-5-amine | SMR000590015 | cid_8122161 | phenyl-(3-phenyl-1,2,4-thiadiazol-5-yl)amine
TypeSmall organic molecule
Emp. Form.C14H11N3S
Mol. Mass.253.322
SMILESN(c1nc(ns1)-c1ccccc1)c1ccccc1
Structure
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