Reaction Details |
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Target | Ubiquitin-conjugating enzyme E2 N |
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Ligand | BDBM50073568 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay |
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IC50 | 1496±84 nM |
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Citation | PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay(2011)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Ubiquitin-conjugating enzyme E2 N |
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Name: | Ubiquitin-conjugating enzyme E2 N |
Synonyms: | BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N |
Type: | PROTEIN |
Mol. Mass.: | 17137.61 |
Organism: | Homo sapiens (Human) |
Description: | EBI_101440 |
Residue: | 152 |
Sequence: | MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
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BDBM50073568 |
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n/a |
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Name | BDBM50073568 |
Synonyms: | 6,7-Dimethoxy-2-piperazin-1-yl-quinazolin-4-ylamine | Aminodimethoxyquinazolinylpiperazine (piperazine derivative of terazosin) | CHEMBL1226 | cid_616267 |
Type | Small organic molecule |
Emp. Form. | C14H19N5O2 |
Mol. Mass. | 289.333 |
SMILES | COc1cc2nc(nc(N)c2cc1OC)N1CCNCC1 |
Structure |
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