Reaction Details |
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Target | Ubiquitin-conjugating enzyme E2 N |
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Ligand | BDBM79314 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay |
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IC50 | 15566±380 nM |
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Citation | PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay(2011)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Ubiquitin-conjugating enzyme E2 N |
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Name: | Ubiquitin-conjugating enzyme E2 N |
Synonyms: | BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N |
Type: | PROTEIN |
Mol. Mass.: | 17137.61 |
Organism: | Homo sapiens (Human) |
Description: | EBI_101440 |
Residue: | 152 |
Sequence: | MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
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BDBM79314 |
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n/a |
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Name | BDBM79314 |
Synonyms: | 6-[2-(4-methyl-1-piperazinyl)-4-pyridinyl]-8-quinolinol | 6-[2-(4-methylpiperazin-1-yl)pyridin-4-yl]quinolin-8-ol | 6-[2-(4-methylpiperazino)-4-pyridyl]quinolin-8-ol | MLS002391557 | SMR001355525 | cid_44142411 |
Type | Small organic molecule |
Emp. Form. | C19H20N4O |
Mol. Mass. | 320.3883 |
SMILES | CN1CCN(CC1)c1cc(ccn1)-c1cc(O)c2ncccc2c1 |
Structure |
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