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TargetX-box-binding protein 1
LigandBDBM68155
Substrate/Competitorn/a
Meas. Tech.XBP1 DR counterscreen for CHOP
IC50 10000±n/a nM
Citation PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
X-box-binding protein 1
Name:X-box-binding protein 1
Synonyms:TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:Enzyme Catalytic Domain
Mol. Mass.:28704.14
Organism:Homo sapiens (Human)
Description:gi_47678753
Residue:261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARK
RQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLR
EKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQL
SPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVP
YQPPFLCQWGRHQPSWKPLMN
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BDBM68155
n/a
NameBDBM68155
Synonyms:MLS001005764 | SMR000384079 | cid_16196355 | nitric acid;2-[(1-phenyl-3-thiophen-2-yl-4-pyrazolyl)methylideneamino]guanidine | nitric acid;2-[(1-phenyl-3-thiophen-2-yl-pyrazol-4-yl)methylideneamino]guanidine | nitric acid;2-[(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)methylideneamino]guanidine | nitric acid;2-[(E)-[1-phenyl-3-(2-thienyl)pyrazol-4-yl]methyleneamino]guanidine | nitric acid;2-[[1-phenyl-3-(2-thienyl)pyrazol-4-yl]methyleneamino]guanidine
TypeSmall organic molecule
Emp. Form.C15H14N6S
Mol. Mass.310.377
SMILES[#7]\[#6](-[#7])=[#7]\[#7]=[#6]-c1cn(nc1-c1cccs1)-c1ccccc1 |w:4.3|
Structure
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