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TargetDNA damage-inducible transcript 3 protein
LigandBDBM67862
Substrate/Competitorn/a
Meas. Tech.CHOP dose-response primary assay
IC50<160±n/a nM
Citation PubChem, PC CHOP dose-response primary assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
DNA damage-inducible transcript 3 protein
Name:DNA damage-inducible transcript 3 protein
Synonyms:Chop | Chop10 | DDIT3_MOUSE | Ddit3 | Gadd153
Type:Enzyme Catalytic Domain
Mol. Mass.:19175.17
Organism:Mus musculus
Description:gi_160707929
Residue:168
Sequence:
MAAESLPFTLETVSSWELEAWYEDLQEVLSSDEIGGTYISSPGNEEEESKTFTTLDPASL
AWLTEEPGPTEVTRTSQSPRSPDSSQSSMAQEEEEEEQGRTRKRKQSGQCPARPGKQRMK
EKEQENERKVAQLAEENERLKQEIERLTREVETTRRALIDRMVSLHQA
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  Blast E-value cutoff:
BDBM67862
n/a
NameBDBM67862
Synonyms:1-(2-chlorobenzyl)-N-[5-(1-ethylpropyl)-1,3,4-thiadiazol-2-yl]-3,5-dimethyl-pyrazole-4-carboxamide | 1-[(2-chlorophenyl)methyl]-3,5-dimethyl-N-(5-pentan-3-yl-1,3,4-thiadiazol-2-yl)-4-pyrazolecarboxamide | 1-[(2-chlorophenyl)methyl]-3,5-dimethyl-N-(5-pentan-3-yl-1,3,4-thiadiazol-2-yl)pyrazole-4-carboxamide | MLS000568058 | SMR000154389 | cid_2550604
TypeSmall organic molecule
Emp. Form.C20H24ClN5OS
Mol. Mass.417.955
SMILESCCC(CC)c1nnc(NC(=O)c2c(C)nn(Cc3ccccc3Cl)c2C)s1
Structure
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