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TargetDNA damage-inducible transcript 3 protein
LigandBDBM68113
Substrate/Competitorn/a
Meas. Tech.CHOP dose-response primary assay
IC50>10000±n/a nM
Citation PubChem, PC CHOP dose-response primary assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
DNA damage-inducible transcript 3 protein
Name:DNA damage-inducible transcript 3 protein
Synonyms:Chop | Chop10 | DDIT3_MOUSE | Ddit3 | Gadd153
Type:Enzyme Catalytic Domain
Mol. Mass.:19175.17
Organism:Mus musculus
Description:gi_160707929
Residue:168
Sequence:
MAAESLPFTLETVSSWELEAWYEDLQEVLSSDEIGGTYISSPGNEEEESKTFTTLDPASL
AWLTEEPGPTEVTRTSQSPRSPDSSQSSMAQEEEEEEQGRTRKRKQSGQCPARPGKQRMK
EKEQENERKVAQLAEENERLKQEIERLTREVETTRRALIDRMVSLHQA
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM68113
n/a
NameBDBM68113
Synonyms:2-[3-(4-methylphenyl)-1-(2-thienylcarbonyl)-4,5-dihydro-1H-pyrazol-5-yl]phenol | MLS000690759 | SMR000301193 | [3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-thiophen-2-yl-methanone | [3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-thiophen-2-ylmethanone | [5-(2-hydroxyphenyl)-3-(p-tolyl)-2-pyrazolin-1-yl]-(2-thienyl)methanone | cid_2988713
TypeSmall organic molecule
Emp. Form.C21H18N2O2S
Mol. Mass.362.445
SMILESCc1ccc(cc1)C1=NN(C(C1)c1ccccc1O)C(=O)c1cccs1 |t:8|
Structure
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