| Reaction Details |
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 | Report a problem with these data |
| Target | Bcl-2-related protein A1 |
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| Ligand | BDBM78578 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen |
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| IC50 | 3320±239 nM |
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| Citation |  PubChem, PC Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Bcl-2-related protein A1 |
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| Name: | Bcl-2-related protein A1 |
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| Synonyms: | A1 | A1-A | B-cell leukemia/lymphoma 2 related protein A1a | B2LA1_MOUSE | Bcl2a1 | Bcl2a1a | Bfl-1 | Bfl1 | Hemopoietic-specific early response protein | Protein BFL-1 |
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| Type: | Apoptosis regulator protein |
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| Mol. Mass.: | 19909.74 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | gi_11024684 |
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| Residue: | 172 |
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| Sequence: | MAESELMHIHSLAEHYLQYVLQVPAFESAPSQACRVLQRVAFSVQKEVEKNLKSYLDDFH
VESIDTARIIFNQVMEKEFEDGIINWGRIVTIFAFGGVLLKKLPQEQIALDVCAYKQVSS
FVAEFIMNNTGEWIRQNGGWEDGFIKKFEPKSGWLTFLQMTGQIWEMLFLLK
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| BDBM78578 |
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| n/a |
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| Name | BDBM78578 |
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| Synonyms: | (E)-3-[3-[(2-bromanyl-4-chloranyl-phenoxy)methyl]-4-methoxy-phenyl]-N-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide | (E)-3-[3-[(2-bromo-4-chloro-phenoxy)methyl]-4-methoxy-phenyl]-N-(1,3,5-trimethylpyrazol-4-yl)acrylamide | (E)-3-[3-[(2-bromo-4-chlorophenoxy)methyl]-4-methoxyphenyl]-N-(1,3,5-trimethyl-4-pyrazolyl)-2-propenamide | (E)-3-[3-[(2-bromo-4-chlorophenoxy)methyl]-4-methoxyphenyl]-N-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide | 3-{3-[(2-bromo-4-chlorophenoxy)methyl]-4-methoxyphenyl}-N-(1,3,5-trimethyl-1H-pyrazol-4-yl)acrylamide | MLS000548222 | SMR000115070 | cid_5430631 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H23BrClN3O3 |
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| Mol. Mass. | 504.804 |
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| SMILES | COc1ccc(\C=C\C(=O)Nc2c(C)nn(C)c2C)cc1COc1ccc(Cl)cc1Br |
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| Structure | 
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