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TargetBcl-2-related protein A1
LigandBDBM78808
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen
IC50 5200±360 nM
Citation PubChem, PC Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Bcl-2-related protein A1
Name:Bcl-2-related protein A1
Synonyms:A1 | A1-A | B-cell leukemia/lymphoma 2 related protein A1a | B2LA1_MOUSE | Bcl2a1 | Bcl2a1a | Bfl-1 | Bfl1 | Hemopoietic-specific early response protein | Protein BFL-1
Type:Apoptosis regulator protein
Mol. Mass.:19909.74
Organism:Mus musculus (Mouse)
Description:gi_11024684
Residue:172
Sequence:
MAESELMHIHSLAEHYLQYVLQVPAFESAPSQACRVLQRVAFSVQKEVEKNLKSYLDDFH
VESIDTARIIFNQVMEKEFEDGIINWGRIVTIFAFGGVLLKKLPQEQIALDVCAYKQVSS
FVAEFIMNNTGEWIRQNGGWEDGFIKKFEPKSGWLTFLQMTGQIWEMLFLLK
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BDBM78808
n/a
NameBDBM78808
Synonyms:2-[4-[2-(4-fluorophenyl)sulfanylethyl]pyridin-1-ium-1-yl]-1-phenyl-ethanone;bromide | 2-[4-[2-(4-fluorophenyl)sulfanylethyl]pyridin-1-ium-1-yl]-1-phenylethanone;bromide | 2-[4-[2-[(4-fluorophenyl)thio]ethyl]-1-pyridin-1-iumyl]-1-phenylethanone;bromide | 2-[4-[2-[(4-fluorophenyl)thio]ethyl]pyridin-1-ium-1-yl]-1-phenyl-ethanone;bromide | 4-{2-[(4-fluorophenyl)thio]ethyl}-1-(2-oxo-2-phenylethyl)pyridinium | MLS000722811 | SMR000304807 | cid_2827177
TypeSmall organic molecule
Emp. Form.C21H19FNOS
Mol. Mass.352.445
SMILESFc1ccc(SCCc2cc[n+](CC(=O)c3ccccc3)cc2)cc1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: