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TargetBcl-2-related protein A1
LigandBDBM79333
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen
IC50 7000±378 nM
Citation PubChem, PC Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Bcl-2-related protein A1
Name:Bcl-2-related protein A1
Synonyms:A1 | A1-A | B-cell leukemia/lymphoma 2 related protein A1a | B2LA1_MOUSE | Bcl2a1 | Bcl2a1a | Bfl-1 | Bfl1 | Hemopoietic-specific early response protein | Protein BFL-1
Type:Apoptosis regulator protein
Mol. Mass.:19909.74
Organism:Mus musculus (Mouse)
Description:gi_11024684
Residue:172
Sequence:
MAESELMHIHSLAEHYLQYVLQVPAFESAPSQACRVLQRVAFSVQKEVEKNLKSYLDDFH
VESIDTARIIFNQVMEKEFEDGIINWGRIVTIFAFGGVLLKKLPQEQIALDVCAYKQVSS
FVAEFIMNNTGEWIRQNGGWEDGFIKKFEPKSGWLTFLQMTGQIWEMLFLLK
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BDBM79333
n/a
NameBDBM79333
Synonyms:MLS002391554 | SMR001355522 | [4-(8-hydroxy-6-quinolinyl)phenyl]-(1-piperazinyl)methanone;2,2,2-trifluoroacetic acid | [4-(8-hydroxy-6-quinolyl)phenyl]-piperazino-methanone;2,2,2-trifluoroacetic acid | [4-(8-hydroxyquinolin-6-yl)phenyl]-piperazin-1-ylmethanone;2,2,2-trifluoroacetic acid | [4-(8-oxidanylquinolin-6-yl)phenyl]-piperazin-1-yl-methanone;2,2,2-tris(fluoranyl)ethanoic acid | cid_44143204
TypeSmall organic molecule
Emp. Form.C20H19N3O2
Mol. Mass.333.3838
SMILESOc1cc(cc2cccnc12)-c1ccc(cc1)C(=O)N1CCNCC1
Structure
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