Reaction Details |
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Target | C-C chemokine receptor type 6 |
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Ligand | BDBM49662 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay |
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IC50 | 552±n/a nM |
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Citation | PubChem, PC Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay PubChem Bioassay(2011)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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C-C chemokine receptor type 6 |
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Name: | C-C chemokine receptor type 6 |
Synonyms: | C-C chemokine receptor type 6 | C-C chemokine receptor type 6 (CCR6) | CCR6 | CCR6_HUMAN | CKRL3 | CMKBR6 | GPR29 | STRL22 |
Type: | Enzyme |
Mol. Mass.: | 42510.84 |
Organism: | Homo sapiens (Human) |
Description: | P51684 |
Residue: | 374 |
Sequence: | MSGESMNFSDVFDSSEDYFVSVNTSYYSVDSEMLLCSLQEVRQFSRLFVPIAYSLICVFG
LLGNILVVITFAFYKKARSMTDVYLLNMAIADILFVLTLPFWAVSHATGAWVFSNATCKL
LKGIYAINFNCGMLLLTCISMDRYIAIVQATKSFRLRSRTLPRSKIICLVVWGLSVIISS
STFVFNQKYNTQGSDVCEPKYQTVSEPIRWKLLMLGLELLFGFFIPLMFMIFCYTFIVKT
LVQAQNSKRHKAIRVIIAVVLVFLACQIPHNMVLLVTAANLGKMNRSCQSEKLIGYTKTV
TEVLAFLHCCLNPVLYAFIGQKFRNYFLKILKDLWCVRRKYKSSGFSCAGRYSENISRQT
SETADNDNASSFTM
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BDBM49662 |
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n/a |
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Name | BDBM49662 |
Synonyms: | MLS000335562 | N-(1H-benzimidazol-2-yl)-3-methyl-1-benzofuran-2-carboxamide | N-(1H-benzimidazol-2-yl)-3-methyl-2-benzofurancarboxamide | N-(1H-benzimidazol-2-yl)-3-methyl-coumarilamide | SMR000253316 | cid_2117785 |
Type | Small organic molecule |
Emp. Form. | C17H13N3O2 |
Mol. Mass. | 291.304 |
SMILES | Cc1c(oc2ccccc12)C(=O)Nc1nc2ccccc2[nH]1 |
Structure |
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