| Reaction Details |
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 | Report a problem with these data |
| Target | cAMP-dependent protein kinase type II-beta regulatory subunit |
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| Ligand | BDBM81294 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R2B (PKA-R2B) complex |
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| EC50 | 66909±n/a nM |
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| Citation |  PubChem, PC Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R2B (PKA-R2B) complex PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| cAMP-dependent protein kinase type II-beta regulatory subunit |
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| Name: | cAMP-dependent protein kinase type II-beta regulatory subunit |
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| Synonyms: | KAP3_HUMAN | PRKAR2B |
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| Type: | PROTEIN |
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| Mol. Mass.: | 46282.41 |
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| Organism: | Homo sapiens (Human) |
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| Description: | EBI_11972 |
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| Residue: | 418 |
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| Sequence: | MSIEIPAGLTELLQGFTVEVLRHQPADLLEFALQHFTRLQQENERKGTARFGHEGRTWGD
LGAAAGGGTPSKGVNFAEEPMQSDSEDGEEEEAAPADAGAFNAPVINRFTRRASVCAEAY
NPDEEEDDAESRIIHPKTDDQRNRLQEACKDILLFKNLDPEQMSQVLDAMFEKLVKDGEH
VIDQGDDGDNFYVIDRGTFDIYVKCDGVGRCVGNYDNRGSFGELALMYNTPRAATITATS
PGALWGLDRVTFRRIIVKNNAKKRKMYESFIESLPFLKSLEFSERLKVVDVIGTKVYNDG
EQIIAQGDSADSFFIVESGEVKITMKRKGKSEVEENGAVEIARCSRGQYFGELALVTNKP
RAASAHAIGTVKCLAMDVQAFERLLGPCMEIMKRNIATYEEQLVALFGTNMDIVEPTA
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| BDBM81294 |
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| n/a |
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| Name | BDBM81294 |
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| Synonyms: | 3-[(2,4-dichlorobenzyl)sulfanyl]-2-thiophenecarboxylic acid | 3-[(2,4-dichlorobenzyl)thio]-2-thenoic acid | 3-[(2,4-dichlorophenyl)methylsulfanyl]thiophene-2-carboxylic acid | 3-[(2,4-dichlorophenyl)methylthio]-2-thiophenecarboxylic acid | MLS000328052 | SMR000168585 | cid_1480284 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H8Cl2O2S2 |
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| Mol. Mass. | 319.227 |
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| SMILES | OC(=O)c1sccc1SCc1ccc(Cl)cc1Cl |
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| Structure | 
|
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