Search and Browse
Download
Enter Data
| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | cAMP-dependent protein kinase type I-alpha regulatory subunit | ||
| Ligand | BDBM66980 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Counterscreen for activators of the Protein Kinase A-R2B (PKA-R2B) complex | ||
| EC50 | 6700±n/a nM | ||
| Citation |  PubChem, PC Counterscreen for activators of the Protein Kinase A-R2B (PKA-R2B) complex: fluorescence polarization-based biochemical high throughput dose response assay to identify activators of the Protein Kinase A-R1A (PKA-R1A) complex PubChem Bioassay(2011)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| cAMP-dependent protein kinase type I-alpha regulatory subunit | |||
| Name: | cAMP-dependent protein kinase type I-alpha regulatory subunit | ||
| Synonyms: | KAP0_BOVIN | PRKAR1A | cAMP-dependent protein kinase | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 42885.14 | ||
| Organism: | Bos taurus | ||
| Description: | gi_115496662 | ||
| Residue: | 380 | ||
| Sequence: |
| ||
| BDBM66980 | |||
| n/a | |||
| Name | BDBM66980 | ||
| Synonyms: | Bucladesine sodium salt | MLS002154012 | SMR001233340 | cid_24871279 | sodium;[(4aS,5R,6R,7aR)-6-[6-(butanoylamino)purin-9-yl]-2-oxidanidyl-2-oxidanylidene-4a,5,6,7a-tetrahydro-4H-furo[2,3-d][1,3,2]dioxaphosphinin-5-yl] butanoate;hydrate | sodium;[(4aS,5R,6R,7aR)-6-[6-(butanoylamino)purin-9-yl]-2-oxido-2-oxo-4a,5,6,7a-tetrahydro-4H-furo[2,3-d][1,3,2]dioxaphosphinin-5-yl] butanoate;hydrate | sodium;butanoic acid [(4aS,5R,6R,7aR)-2-oxido-2-oxo-6-[6-(1-oxobutylamino)-9-purinyl]-4a,5,6,7a-tetrahydro-4H-furo[2,3-d][1,3,2]dioxaphosphorin-5-yl] ester;hydrate | sodium;butyric acid [(4aS,5R,6R,7aR)-6-(6-butyramidopurin-9-yl)-2-keto-2-oxido-4a,5,6,7a-tetrahydro-4H-furo[2,3-d][1,3,2]dioxaphosphorin-5-yl] ester;hydrate | ||
| Type | Small organic molecule | ||
| Emp. Form. | C18H23N5O8P | ||
| Mol. Mass. | 468.3782 | ||
| SMILES | CCCC(=O)Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2OP([O-])(=O)OC[C@H]2[C@H]1OC(=O)CCC | ||
| Structure | 
| ||