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TargetProtachykinin-1
LigandBDBM50010685
Substrate/Competitorn/a
Ki>10000±n/a nM
CommentsPDSP_664
Citation Mottola, DMBrewster, WKCook, LLNichols, DEMailman, RB Dihydrexidine, a novel full efficacy D1 dopamine receptor agonist. J Pharmacol Exp Ther262:383-93 (1992) [PubMed]
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Protachykinin-1
Name:Protachykinin-1
Synonyms:Nka | Nkna | Protachykinin-1 | Substance K | Substance P | TKN1_RAT | Tac1 | Tac2
Type:Enzyme Catalytic Domain
Mol. Mass.:15007.06
Organism:RAT
Description:Substance K 0 RAT::P06767
Residue:130
Sequence:
MKILVAVAVFFLVSTQLFAEEIGANDDLNYWSDWSDSDQIKEAMPEPFEHLLQRIARRPK
PQQFFGLMGKRDADSSIEKQVALLKALYGHGQISHKRHKTDSFVGLMGKRALNSVAYERS
AMQNYERRRK
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  Blast E-value cutoff:
BDBM50010685
n/a
NameBDBM50010685
Synonyms:(+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahydrobenzo[a]phenanthridine | (6aR,12bR)-5,6,6a,7,8,12b-Hexahydro-benzo[a]phenanthridine-10,11-diol | 5,6,6a,7,8,12b-Hexahydro-benzo[a]phenanthridine-10,11-diol | CHEMBL43345 | Dihydrexidine, DHX
TypeSmall organic molecule
Emp. Form.C17H17NO2
Mol. Mass.267.3224
SMILESOc1cc2CC[C@H]3NCc4ccccc4[C@H]3c2cc1O
Structure
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