Reaction Details |
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Target | Beta-arrestin-2 |
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Ligand | BDBM81875 |
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Substrate/Competitor | n/a |
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Ki | 154.88±n/a nM |
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Comments | PDSP_831 |
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Citation | Wong, DT; Threlkeld, PG; Robertson, DW Affinities of fluoxetine, its enantiomers, and other inhibitors of serotonin uptake for subtypes of serotonin receptors. Neuropsychopharmacology5:43-7 (1991) [PubMed] |
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More Info.: | Get all data from this article |
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Beta-arrestin-2 |
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Name: | Beta-arrestin-2 |
Synonyms: | 5-HT2C | ARRB2 | ARRB2_BOVIN | Beta-arrestin-2 | HTR2C |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 47232.00 |
Organism: | Beef |
Description: | 5-HT2C HTR2C Beef::P32120 |
Residue: | 420 |
Sequence: | MGEKPGTRVFKKSSPNCKLTVYLGKRDFVDHLDKVDPVDGVVLVDPDYLKDRKVFVTLTC
AFRYGREDLDVLGLSFRKDLFIANYQAFPPTPNPPRPPTRLQERLLRKLGQHAHPFFFTI
PQNLPCSVTLQPGPEDTGKACGVDFEIRAFCAKSLEEKSHKRNSVRLVIRKVQFAPEKPG
PQPSAETTRHFLMSDRSLHLEASLDKELYYHGEPLNVNVHVTNNSTKTVKKIKVSVRQYA
DICLFSTAQYKCPVAQVEQDDQVSPSSTFCKVYTITPLLSNNREKRGLALDGKLKHEDTN
LASSTIVKEGANKEVLGILVSYRVKVKLVVSRGGDVSVELPFVLMHPKPHDHIALPRPQS
AATHPPTLLPSAVPETDAPVDTNLIEFETNYATDDDIVFEDFARLRLKGLKDEDYDDQFC
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BDBM81875 |
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n/a |
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Name | BDBM81875 |
Synonyms: | Fluoxetine-R-(-) |
Type | n/a |
Emp. Form. | C17H18F3NO |
Mol. Mass. | 309.3261 |
SMILES | CNCC[C@H](Oc1ccc(cc1)C(F)(F)F)c1ccccc1 |
Structure |
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