| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM81925 |
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| Substrate/Competitor | n/a |
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| Ki | 2.9±n/a nM |
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| Comments | PDSP_2952 |
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| Citation |  Klotz, KN; Vogt, H; Tawfik-Schlieper, H Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling. Naunyn Schmiedebergs Arch Pharmacol343:196-201 (1991) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | AA3R_SHEEP | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADENOSINE A3 | ADORA1 | ADORA3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36152.74 |
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| Organism: | Sheep |
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| Description: | ADENOSINE A1 ADORA1 Sheep::P35342 |
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| Residue: | 317 |
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| Sequence: | MPVNSTAVSWTSVTYITVEILIGLCAIVGNVLVIWVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVISLGVTIHFYSCLFMTCLMLIFTHASIMSLLAIAVDRYLRVKLTVRYRR
VTTQRRIWLALGLCWLVSFLVGLTPMFGWNMKLSSADENLTFLPCRFRSVMRMDYMVYFS
FFLWILVPLVVMCAIYFDIFYIIRNRLSQSFSGSRETGAFYGREFKTAKSLLLVLFLFAL
CWLPLSIINCILYFDGQVPQTVLYLGILLSHANSMMNPIVYAYKIKKFKETYLLILKACV
MCQPSKSMDPSTEQTSE
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| BDBM81925 |
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| n/a |
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| Name | BDBM81925 |
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| Synonyms: | 8-Cyclopentyl-1,3-dimethyl-3,7-dihydro-purine-2,6-dione | 8-Cyclopentyltheophylline (CPT) | CAS_1917 | CHEMBL106265 | CPT | NSC_1917 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H16N4O2 |
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| Mol. Mass. | 248.281 |
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| SMILES | Cn1c2nc([nH]c2c(=O)n(C)c1=O)C1CCCC1 |
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| Structure | 
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