| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Adenosine receptor A3 |
|---|
| Ligand | BDBM50008415 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 0.98±n/a nM |
|---|
| Comments | PDSP_2055 |
|---|
| Citation |  Klotz, KN; Vogt, H; Tawfik-Schlieper, H Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling. Naunyn Schmiedebergs Arch Pharmacol343:196-201 (1991) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Adenosine receptor A3 |
|---|
| Name: | Adenosine receptor A3 |
|---|
| Synonyms: | AA3R_SHEEP | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADENOSINE A3 | ADORA1 | ADORA3 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 36152.74 |
|---|
| Organism: | Sheep |
|---|
| Description: | ADENOSINE A1 ADORA1 Sheep::P35342 |
|---|
| Residue: | 317 |
|---|
| Sequence: | MPVNSTAVSWTSVTYITVEILIGLCAIVGNVLVIWVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVISLGVTIHFYSCLFMTCLMLIFTHASIMSLLAIAVDRYLRVKLTVRYRR
VTTQRRIWLALGLCWLVSFLVGLTPMFGWNMKLSSADENLTFLPCRFRSVMRMDYMVYFS
FFLWILVPLVVMCAIYFDIFYIIRNRLSQSFSGSRETGAFYGREFKTAKSLLLVLFLFAL
CWLPLSIINCILYFDGQVPQTVLYLGILLSHANSMMNPIVYAYKIKKFKETYLLILKACV
MCQPSKSMDPSTEQTSE
|
|
|
|---|
| BDBM50008415 |
|---|
| n/a |
|---|
| Name | BDBM50008415 |
|---|
| Synonyms: | 2-(2-Chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | 2-[2-chloro-6-(cyclopentylamino)-9H-purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | CCPA |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H20ClN5O4 |
|---|
| Mol. Mass. | 369.803 |
|---|
| SMILES | OCC1OC(C(O)C1O)n1cnc2c(NC3CCCC3)nc(Cl)nc12 |
|---|
| Structure | 
|
|---|
Search and Browse
