| Reaction Details |
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 | Report a problem with these data |
| Target | Protachykinin-1 |
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| Ligand | BDBM81942 |
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| Substrate/Competitor | n/a |
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| Ki | 4.6±n/a nM |
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| Comments | PDSP_1774 |
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| Citation |  Burcher, E; Buck, SH; Lovenberg, W; O'Donohue, TL Characterization and autoradiographic localization of multiple tachykinin binding sites in gastrointestinal tract and bladder. J Pharmacol Exp Ther236:819-31 (1986) [PubMed] |
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| More Info.: | Get all data from this article |
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| Protachykinin-1 |
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| Name: | Protachykinin-1 |
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| Synonyms: | Nka | Nkna | Protachykinin-1 | Substance K | Substance P | TKN1_RAT | Tac1 | Tac2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 15007.06 |
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| Organism: | RAT |
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| Description: | Substance K 0 RAT::P06767 |
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| Residue: | 130 |
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| Sequence: | MKILVAVAVFFLVSTQLFAEEIGANDDLNYWSDWSDSDQIKEAMPEPFEHLLQRIARRPK
PQQFFGLMGKRDADSSIEKQVALLKALYGHGQISHKRHKTDSFVGLMGKRALNSVAYERS
AMQNYERRRK
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| BDBM81942 |
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| n/a |
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| Name | BDBM81942 |
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| Synonyms: | CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | Substance K |
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| Type | Small organic molecule |
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| Emp. Form. | C50H80N14O14S |
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| Mol. Mass. | 1133.321 |
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| SMILES | CSCCC(NC(=O)C(CC(C)C)NC(=O)CNC(=O)C(NC(=O)C(Cc1ccccc1)NC(=O)C(CO)NC(=O)C(CC(O)=O)NC(=O)C(NC(=O)C(CCCCN)NC(=O)C(N)Cc1cnc[nH]1)C(C)O)C(C)C)C(N)=O |
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| Structure | 
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