| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
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| Ligand | BDBM50002051 |
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| Substrate/Competitor | n/a |
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| Ki | 141±n/a nM |
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| Comments | PDSP_643 |
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| Citation |  Mendelsohn, LG; Kalra, V; Johnson, BG; Kerchner, GA Sigma opioid receptor: characterization and co-identity with the phencyclidine receptor. J Pharmacol Exp Ther233:597-602 (1985) [PubMed] |
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| More Info.: | Get all data from this article |
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| Sigma non-opioid intracellular receptor 1 |
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| Name: | Sigma non-opioid intracellular receptor 1 |
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| Synonyms: | Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25266.54 |
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| Organism: | RAT |
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| Description: | Q9R0C9 |
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| Residue: | 223 |
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| Sequence: | MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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| BDBM50002051 |
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| n/a |
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| Name | BDBM50002051 |
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| Synonyms: | (+/-)-(2RS)-2-[(4RS)-2,2-Diphenyl-1,3-dioxolan-4-yl]piperidine | (+/-)-(2RS)-2-[(4SR)-2,2-diphenyl-1,3-dioxolan-4-yl]piperidine | (Dexoxadrol)2-(2,2-Diphenyl-[1,3]dioxolan-4-yl)-piperidine | CHEMBL26479 | Dexoxadrol |
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| Type | Small organic molecule |
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| Emp. Form. | C20H23NO2 |
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| Mol. Mass. | 309.4021 |
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| SMILES | C1OC(OC1C1CCCCN1)(c1ccccc1)c1ccccc1 |
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| Structure | 
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