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TargetCholinergic, muscarinic
LigandBDBM50004665
Substrate/Competitorn/a
Ki 214±n/a nM
CommentsPDSP_1426
Citation Bloom JWHalonen MLawrence LJRould ESeaver NAYamamura HI Characterization of high affinity [3H]pirenzepine and (-)-[3H] quinuclidinyl benzilate binding to muscarinic cholinergic receptors in rabbit peripheral lung. J Pharmacol Exp Ther 240:51-8 (1987) [PubMed]
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Cholinergic, muscarinic
Name:Cholinergic, muscarinic
Synonyms:Beta-arrestin-1 | OPIATE Delta | PAF Platelet activating factor
Type:Enzyme Catalytic Domain
Mol. Mass.:46360.54
Organism:RABBIT
Description:Cholinergic, muscarinic 0 RABBIT::Q95223
Residue:410
Sequence:
MGDKGTRVFKKASPNGKLTVYLGKRGFVDHIDLVDPVDGVVLVDPEYLKERRVYVTLTCA
FRYGREDLDVLGLTFRKDLFVANVQSFPPAPEDKKPLTRLQERLIKKLGEHAYPFTFEIP
PKLPCSVTLQPGPEDTGKACGVDYEVKAFCAENLEEKIHKRNSVRLVIRKVQYAPERPGP
HPTAETTRLFLMSDKPLHLEASLDKEIYYHGEPIIVNVHVTNNTNKTVKKIKISVRQYAD
ICLFNTAQYKCPVAMEEADDTVAPSSTFCKVYTLTPFLANNREKRGLALDGKLKHEDTNL
ASSTLMREGANREILGIIVSYKVKVKLVVSRGGDVAVELPFTLMHPKPKEEPPHREVPEN
ETPVDTNLIELDTNDDDIVFEDFARQRLKGMKDDKEEEDDVTGSPRLNDR
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BDBM50004665
n/a
NameBDBM50004665
Synonyms:(oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | 1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | 1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one (oxotremorphine) | 1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one(Oxotremorine) | 1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidinium | CHEMBL7634 | Oxotremorine | Oxotremorine1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | cid_4630
TypeSmall organic molecule
Emp. Form.C12H18N2O
Mol. Mass.206.2841
SMILESO=C1CCCN1CC#CCN1CCCC1
Structure
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