Reaction Details | |||
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Target | Histamine H1 receptor | ||
Ligand | BDBM50005548 | ||
Substrate/Competitor | n/a | ||
Ki | 2700±n/a nM | ||
Comments | PDSP_1347 | ||
Citation | Kanba, S; Richelson, E Histamine H1 receptors in human brain labelled with [3H]doxepin. Brain Res304:1-7 (1984) [PubMed] Article | ||
More Info.: | Get all data from this article | ||
Histamine H1 receptor | |||
Name: | Histamine H1 receptor | ||
Synonyms: | H1R | HH1R | HISTAMINE H1 | HRH1 | HRH1_HUMAN | ||
Type: | G Protein-Coupled Receptor (GPCR) | ||
Mol. Mass.: | 55808.72 | ||
Organism: | Homo sapiens (Human) | ||
Description: | Cell pellets from SK-N-MC cells transfected with human H1 receptor were used in binding assay. | ||
Residue: | 487 | ||
Sequence: |
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BDBM50005548 | |||
n/a | |||
Name | BDBM50005548 | ||
Synonyms: | (+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | (+/-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | (-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | (Nomifensine) 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine (Nomifensine) | 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine(Nomifensine) | 2-methyl-4-phenyl-1,2,3,4-tetrahydroisoquinolin-8-amine | CHEMBL273575 | NOMIFENSINE | NOMIFENSINE2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | ||
Type | Small organic molecule | ||
Emp. Form. | C16H18N2 | ||
Mol. Mass. | 238.3275 | ||
SMILES | CN1CC(c2ccccc2)c2cccc(N)c2C1 | ||
Structure |