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TargetSomatostatin receptor type 1
LigandBDBM82255
Substrate/Competitorn/a
Ki>10000±n/a nM
CommentsPDSP_1295
Citation Rossowski, WJGu, ZFAkarca, USJensen, RTCoy, DH Characterization of somatostatin receptor subtypes controlling rat gastric acid and pancreatic amylase release. Peptides15:1421-4 (1994) [PubMed]  Article
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Somatostatin receptor type 1
Name:Somatostatin receptor type 1
Synonyms:SOMATOSTATIN SST1 | SRIF-2 | SS1R | SSR1_RAT | Somatostatin receptor | Somatostatin receptor type 1 | Sstr1
Type:Enzyme Catalytic Domain
Mol. Mass.:42752.93
Organism:RAT
Description:SOMATOSTATIN SST1 SSTR1 RAT::P28646
Residue:391
Sequence:
MFPNGTAPSPTSSPSSSPGGCGEGVCSRGPGSGAADGMEEPGRNSSQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCASRISTL
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  Blast E-value cutoff:
BDBM82255
n/a
NameBDBM82255
Synonyms:D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12
Typen/a
Emp. Form.C57H69N11O8S2
Mol. Mass.1100.357
SMILESNCCCCC1NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(CSSCC(NC(=O)C(CCCN)NC1=O)C(=O)NCc1cccc2ccccc12)NC(=O)C(N)Cc1ccccc1
Structure
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