| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Melatonin receptor type 1A |
|---|
| Ligand | BDBM50034110 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 0.21±n/a nM |
|---|
| Comments | PDSP_1193 |
|---|
| Citation |  Reppert, SM; Godson, C; Mahle, CD; Weaver, DR; Slaugenhaupt, SA; Gusella, JF Molecular characterization of a second melatonin receptor expressed in human retina and brain: the Mel1b melatonin receptor. Proc Natl Acad Sci U S A92:8734-8 (1995) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Melatonin receptor type 1A |
|---|
| Name: | Melatonin receptor type 1A |
|---|
| Synonyms: | MTNR1A | MTNR1A protein | MTR1A_HUMAN | Mel-1A-R | Mel1a melatonin receptor | Melatonin 1A | Melatonin receptor | Melatonin receptor 1A | Melatonin receptor type 1 (MT1) | Melatonin receptor type 1A |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 39392.94 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P48039 |
|---|
| Residue: | 350 |
|---|
| Sequence: | MQGNGSALPNASQPVLRGDGARPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRN
AGNIFVVSLAVADLVVAIYPYPLVLMSIFNNGWNLGYLHCQVSGFLMGLSVIGSIFNITG
IAINRYCYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFA
QSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRQRVKPDRKPKLKPQDFRNFVTM
FVVFVLFAICWAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNAIIYGLLNQ
NFRKEYRRIIVSLCTARVFFVDSSNDVADRVKWKPSPLMTNNNVVKVDSV
|
|
|
|---|
| BDBM50034110 |
|---|
| n/a |
|---|
| Name | BDBM50034110 |
|---|
| Synonyms: | CHEMBL15060 | Melatonin,2-Phenyl | N-[2-(5-Methoxy-2-phenyl-1H-indol-3-yl)-ethyl]-acetamide |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H20N2O2 |
|---|
| Mol. Mass. | 308.3743 |
|---|
| SMILES | COc1ccc2[nH]c(c(CCNC(C)=O)c2c1)-c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
