| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptides B/W receptor type 1 |
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| Ligand | BDBM21864 |
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| Substrate/Competitor | n/a |
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| Ki | 1226±n/a nM |
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| Comments | PDSP_1287 |
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| Citation |  O'Dowd, BF; Scheideler, MA; Nguyen, T; Cheng, R; Rasmussen, JS; Marchese, A; Zastawny, R; Heng, HH; Tsui, LC; Shi, X The cloning and chromosomal mapping of two novel human opioid-somatostatin-like receptor genes, GPR7 and GPR8, expressed in discrete areas of the brain. Genomics28:84-91 (1995) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Neuropeptides B/W receptor type 1 |
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| Name: | Neuropeptides B/W receptor type 1 |
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| Synonyms: | GPR7 | NPBW1_HUMAN | NPBWR1 | neuropeptides B/W receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36111.82 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_119607128 |
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| Residue: | 328 |
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| Sequence: | MDNASFSEPWPANASGPDPALSCSNASTLAPLPAPLAVAVPVVYAVICAVGLAGNSAVLY
VLLRAPRMKTVTNLFILNLAIADELFTLVLPINIADFLLRQWPFGELMCKLIVAIDQYNT
FSSLYFLTVMSADRYLVVLATAESRRVAGRTYSAARAVSLAVWGIVTLVVLPFAVFARLD
DEQGRRQCVLVFPQPEAFWWRASRLYTLVLGFAIPVSTICVLYTTLLCRLHAMRLDSHAK
ALERAKKRVTFLVVAILAVCLLCWTPYHLSTVVALTTDLPQTPLVIAISYFITSLSYANS
CLNPFLYAFLDASFRRNLRQLITCRAAA
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| BDBM21864 |
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| n/a |
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| Name | BDBM21864 |
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| Synonyms: | (21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5,7,9,15,17,19(25)-heptaene-2,16-diol | (8R)-7-(cyclopropylmethyl)-5,6,7,8,14,14b-hexahydro-4,8-methano[1]benzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol | NALTRINDOLE | [3H]-naltrindole |
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| Type | radiolabeled ligand |
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| Emp. Form. | C26H26N2O3 |
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| Mol. Mass. | 414.4962 |
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| SMILES | [H][C@@]12Cc3ccc(O)c4OC5c6[nH]c7ccccc7c6CC1(O)C5(CCN2CC1CC1)c34 |THB:27:26:21:31.2.3| |
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| Structure | 
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